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Page 1
Trypanocidal potential of synthetic p-aminochalcones: In silico and in vitro evaluation.
Dutra Barroso Gomes N, Paula Magalhães E, Rodrigues Ribeiro L, Cavalcante JW, Morais Gomes Maia M, Cunha da Silva FR, Ali A, Machado Marinho M, Silva Marinho E, Silva Dos Santos H, Costa Martins AM, Róseo Paula Pessoa Bezerra de Menezes R. Dutra Barroso Gomes N, et al. Among authors: paula magalhaes e. Bioorg Chem. 2023 Dec;141:106931. doi: 10.1016/j.bioorg.2023.106931. Epub 2023 Oct 20. Bioorg Chem. 2023. PMID: 37879182
Rational design of a trypanocidal peptide derived from Dinoponera quadriceps venom.
Monteiro ML, Lima DB, Freire KA, Nicolaski Pedron C, Magalhães EP, Silva BP, García-Jareño AB, De Oliveira CS, Nunes JVS, Marinho MM, Menezes RRPPB, Orzaéz M, Oliveira Junior VX, Martins AMC. Monteiro ML, et al. Among authors: magalhaes ep. Eur J Med Chem. 2022 Nov 5;241:114624. doi: 10.1016/j.ejmech.2022.114624. Epub 2022 Jul 31. Eur J Med Chem. 2022. PMID: 35933786
GABAA and serotonergic receptors participation in anxiolytic effect of chalcones in adult zebrafish.
Mendes FRS, da Silva AW, Ferreira MKA, Rebouças EL, Moura Barbosa I, da Rocha MN, Henrique Ferreira Ribeiro W, Menezes RRPPB, Magalhães EP, Marinho EM, Marinho MM, Bandeira PN, de Menezes JESA, Marinho ES, Dos Santos HS. Mendes FRS, et al. Among authors: magalhaes ep. J Biomol Struct Dyn. 2023;41(21):12426-12444. doi: 10.1080/07391102.2023.2167116. Epub 2023 Jan 16. J Biomol Struct Dyn. 2023. PMID: 36644862
Antiparasitary and antiproliferative activities in vitro of a 1,2,4-oxadiazole derivative on Trypanosoma cruzi.
Rocha YM, Magalhães EP, de Medeiros Chaves M, Machado Marinho M, Nascimento E Melo de Oliveira V, Nascimento de Oliveira R, Lima Sampaio T, de Menezes RRPPB, Martins AMC, Nicolete R. Rocha YM, et al. Among authors: magalhaes ep. Parasitol Res. 2022 Jul;121(7):2141-2156. doi: 10.1007/s00436-022-07554-z. Epub 2022 May 25. Parasitol Res. 2022. PMID: 35610523
Chloride substitution on 2-hydroxy-3,4,6-trimethoxyphenylchalcones improves in vitro selectivity on Trypanosoma cruzi strain Y.
Magalhães EP, Gomes NDB, Freitas TA, Silva BP, Ribeiro LR, Ameida-Neto FWQ, Marinho MM, Lima-Neto P, Marinho ES, Santos HSD, Teixeira AMR, Sampaio TL, Menezes RRPPB, Martins AMC. Magalhães EP, et al. Chem Biol Interact. 2022 Jul 1;361:109920. doi: 10.1016/j.cbi.2022.109920. Epub 2022 Apr 21. Chem Biol Interact. 2022. PMID: 35461787
Antiproliferative activity on Trypanosoma cruzi (Y strain) of the triterpene 3β,6β,16β-trihidroxilup-20 (29)-ene isolated from Combretum leprosum.
de Araújo JIF, Aires NL, Almeida-Neto FWQ, Marinho MM, Marinho EM, Paula Magalhães E, de Menezes RRPPB, Sampaio TL, Maria Costa Martins A, Teixeira EH, Rafaela Freitas Dotto A, Amaral WD, Teixeira AMR, de Lima-Neto P, Marinho ES, Dos Santos HS. de Araújo JIF, et al. Among authors: paula magalhaes e. J Biomol Struct Dyn. 2022;40(22):12302-12315. doi: 10.1080/07391102.2021.1970025. Epub 2021 Aug 26. J Biomol Struct Dyn. 2022. PMID: 34436980
Effect from dinoponeratoxin M-PONTXDq3a arginine and lysine substituted analogues against Staphylococcus aureus strains.
Nonato da Silva Júnior P, Serra Nunes JV, Duque BR, Batista Pereira AJ, Magalhães EP, Oliveira CS, Freire KA, Pedron CN, Oliveira VX, Sampaio TL, Costa Martins AM. Nonato da Silva Júnior P, et al. Among authors: magalhaes ep. Toxicon. 2023 Aug 1;231:107190. doi: 10.1016/j.toxicon.2023.107190. Epub 2023 Jun 8. Toxicon. 2023. PMID: 37301297
18 results